SCHEMBL17156366

SCHEMBL17156366

CCOc1nn(-c2ccccn2)c2c1CCN(Cc1ccccc1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.43
MAPT P10636 4/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
C5AR1 P21730 1/20 0.40
LMNA P02545 4/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
MAPK1 P28482 1/20 0.39
MEN1 O00255 1/20 0.38
ADORA1 P30542 1/20 0.38
KMT2A Q03164 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
CLPP Q16740 1/20 0.38
AVPR1A P37288 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391586 0.92 C5AR1 (0.43) HTTMAPTNPC1RAB9AC5AR1
SCHEMBL3390126 0.77 CLPP (0.45) C5AR1CLPPDRD2DRD4DRD3
SCHEMBL23648628 0.75 C5AR1 (0.46) HTTMAPTNPC1RAB9AC5AR1
SCHEMBL29871610 0.75 C5AR1 (0.46) HTTMAPTNPC1RAB9AC5AR1
SCHEMBL3390729 0.74 CLPP (0.46) C5AR1CLPPDRD2DRD4DRD3
SCHEMBL3390016 0.74 CLPP (0.45) C5AR1CLPPDRD2DRD4DRD3
SCHEMBL29871084 0.73 MAPT (0.44) HTTMAPTNPC1RAB9ALMNA
SCHEMBL23648607 0.73 MAPT (0.44) HTTMAPTNPC1RAB9ALMNA
Hydrochloric Acid SCHEMBL23648819 0.73 MAPT (0.43) HTTMAPTNPC1RAB9ALMNA
Hydrochloric Acid SCHEMBL29871578 0.73 MAPT (0.43) HTTMAPTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2929883-A1 Pyrazole derivatives as dihydroorotate dehydrogenase (DHODH) inhibitors INSTITUT PASTEUR (FR) 2015-10-14 EP disclosed