SCHEMBL17166118

SCHEMBL17166118

COC(=O)c1c(F)cccc1CF

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
BDKRB1 P46663 16/20 0.48
KMT2A Q03164 2/20 0.47
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18329438 0.88 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL1070351 0.87 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL19497046 0.86 BDKRB1 (0.49) CA12CA1CA2CA7CA9
SCHEMBL8322933 0.85 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL29026652 0.81 BDKRB1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL22445329 0.81 BDKRB1 (0.44) CA12CA1CA2CA7CA9
SCHEMBL23748265 0.80 MAOB (0.54) BDKRB1KMT2A
SCHEMBL6618372 0.80 HDAC1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL28342751 0.79 PLK1 (0.49) CA12CA1CA2CA7CA9
SCHEMBL16664442 0.79 GAA (0.49) KMT2ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9156791-B2 Pyrazole compounds acting against allergic, immune and inflammatory conditions GLAXO GROUP LIMITED (GB) 2015-10-13 US disclosed