SCHEMBL29026652

SCHEMBL29026652

COC(=O)c1c(F)cccc1CC#N

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 18/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131128 0.83 CA12 (0.44) BDKRB1MEN1KMT2ACA12CA1
SCHEMBL18329438 0.82 CA12 (0.50) BDKRB1KMT2ACA12CA1CA2
SCHEMBL24317461 0.82 CA12 (0.43) BDKRB1MEN1KMT2ACA12CA1
SCHEMBL29026633 0.82 LMNA (0.49) BDKRB1MEN1KMT2ACA12CA1
SCHEMBL19497046 0.81 BDKRB1 (0.49) BDKRB1KMT2ACA12CA1CA2
SCHEMBL17166118 0.81 CA12 (0.48) BDKRB1KMT2ACA12CA1CA2
SCHEMBL8322933 0.80 CA12 (0.47) BDKRB1KMT2ACA12CA1CA2
SCHEMBL29131122 0.79 BDKRB1 (0.38) BDKRB1CA12CA1CA2CA7
SCHEMBL29199348 0.79 BDKRB1 (0.38) BDKRB1MEN1KMT2ACA12CA1
SCHEMBL4968519 0.79 ALDH1A1 (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN claimed
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN disclosed
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-116375704-A KRAS G12C Preparation and application of mutant protein isoquinolinone inhibitor 药雅科技(上海)有限公司 2023-07-04 CN disclosed