SCHEMBL6618372

SCHEMBL6618372

COC(=O)c1c(F)cccc1CCCBr

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
BDKRB1 P46663 15/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
KMT2A Q03164 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322933 0.84 CA12 (0.47) BDKRB1CA12CA1CA2CA7
SCHEMBL18329438 0.81 CA12 (0.50) BDKRB1CA12CA1CA2CA7
SCHEMBL17166118 0.80 CA12 (0.48) BDKRB1CA12CA1CA2CA7
SCHEMBL19497046 0.80 BDKRB1 (0.49) BDKRB1CA12CA1CA2CA7
SCHEMBL1070351 0.77 CA12 (0.61) BDKRB1CA12CA1CA2CA7
SCHEMBL6621914 0.75 ALDH1A1 (0.64) CA1CA2CA9KMT2A
SCHEMBL29026652 0.75 BDKRB1 (0.47) BDKRB1CA12CA1CA2CA7
SCHEMBL22445329 0.75 BDKRB1 (0.44) BDKRB1CA12CA1CA2CA7
SCHEMBL10561912 0.74 CA12 (0.46) HDAC1HDAC6CA12CA1CA2
SCHEMBL27859776 0.74 HDAC1 (0.46) HDAC1HDAC6BDKRB1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683781-B1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE METABASIS THERAPEUTICS INC (US) 2004-04-21 EP disclosed
US-5731432-A Inhibitors of adenosine monophosphate deaminase GENSIA SICOR INC. (US) 1998-03-24 US disclosed
EP-0683781-A4 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE. GENSIA PHARMA (US) 1997-05-28 EP disclosed
EP-0683781-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA PHARMACEUTICALS, INC. (US) 1995-11-29 EP disclosed
WO-1994018200-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA, INC. (US) 1994-08-18 WO disclosed