SCHEMBL17166286

SCHEMBL17166286

COc1cc2oc(-c3ccc(O)cc3)cc(=O)c2c(O)c1-c1cc(-c2cc(=O)c3c(O)cc(O)cc3o2)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 6/20 1.00
MMP3 P08254 1/20 0.79
MMP9 P14780 1/20 0.79
MAPT P10636 6/20 0.68
CYP1B1 Q16678 5/20 0.68
MEN1 O00255 5/20 0.68
KMT2A Q03164 5/20 0.68
CYP1A1 P04798 4/20 0.68
CYP1A2 P05177 4/20 0.68
POLB P06746 4/20 0.68
ABCC1 P33527 3/20 0.68
ALDH1A1 P00352 3/20 0.68
IP6K2 Q9UHH9 4/20 0.65
XDH P47989 2/20 0.65
IPMK Q8NFU5 2/20 0.65
HDAC6 Q9UBN7 2/20 0.65
KDM1A O60341 1/20 0.65
TDP1 Q9NUW8 4/20 0.64
THRB P10828 2/20 0.64
PTPN1 P18031 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17166013 0.94 APP (0.89) APPMMP3MMP9MAPTCYP1B1
SCHEMBL7637240 0.89 APP (0.81) APPMMP3MMP9MAPTCYP1B1
SCHEMBL13672774 0.89 APP (0.80) APPMMP3MMP9MAPTMEN1
Sotetsuflavone SCHEMBL4467051 0.89 APP (0.80) APPMMP3MMP9MAPTCYP1B1
Sotetsuflavone SCHEMBL30646165 0.89 APP (0.80) APPMMP3MMP9MAPTCYP1B1
SCHEMBL30766312 0.88 APP (0.79) APPMMP3MMP9MAPTCYP1B1
Robustaflavone SCHEMBL561807 0.87 APP (0.77) APPMMP3MMP9MAPTCYP1B1
SCHEMBL30799700 0.87 APP (0.83) APPMMP3MMP9MAPTCYP1B1
Robustaflavone SCHEMBL7638211 0.86 APP (0.76) APPMMP3MMP9MAPTCYP1B1
Robustaflavone SCHEMBL7643511 0.86 APP (0.76) APPMMP3MMP9MAPTCYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9155792-B2 RecA inhibitors with antibiotic activity, compositions and methods of use TRUSTEES OF BOSTON UNIVERSITY (US) 2015-10-13 US disclosed