SCHEMBL17166394

SCHEMBL17166394

CC(C)(C)OC(=O)C1CN(Cc2ccccc2)C(Br)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
MAPT P10636 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
ABCB1 P08183 1/20 0.36
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1947707 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL22039863 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL20146480 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL22039864 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL17986811 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL30636976 0.76 MAPT (0.50) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL11197364 0.75 MMP13 (0.53) KMT2AL3MBTL1ALDH1A1TSHRMAPK1
SCHEMBL17166392 0.75 KMT2A (0.42) KMT2AL3MBTL1MAPTALDH1A1JAK2
Hydrochloric Acid SCHEMBL28654829 0.74 MAPT (0.49) KMT2AL3MBTL1PDK1PDK2PDK3
SCHEMBL2342290 0.73 KMT2A (0.45) KMT2AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9156858-B2 Boronic acid derivatives and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2015-10-13 US disclosed