SCHEMBL17169477

SCHEMBL17169477

CC(C)(C)OC(=O)N[C@](C)(c1ccccc1F)[C@@H](F)[C@H](O)C(C)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
AAK1 Q2M2I8 4/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
SCN9A Q15858 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRB2 P47870 1/20 0.33
AKT1 P31749 1/20 0.33
MAPK10 P53779 1/20 0.33
PTPN1 P18031 1/20 0.32
APLNR P35414 1/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
ADRB3 P13945 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18636854 1.00 LMNA (0.40) LMNAPOLBCTSSCTSKAAK1
SCHEMBL17169302 0.83 LMNA (0.36) LMNAPOLBCTSSCTSKAAK1
SCHEMBL18636691 0.82 LMNA (0.33) LMNAPOLBCTSSCTSKAAK1
SCHEMBL17169468 0.80 LMNA (0.39) LMNAPOLBCTSSCTSKAAK1
SCHEMBL21677228 0.80 LMNA (0.39) LMNAPOLBCTSSCTSKAAK1
SCHEMBL18683370 0.80 CTSS (0.40) LMNAPOLBCTSSCTSKAAK1
SCHEMBL18683500 0.80 LMNA (0.39) LMNAPOLBCTSSCTSKAAK1
SCHEMBL18623895 0.79 LMNA (0.38) LMNAPOLBCTSSCTSKAAK1
SCHEMBL18636851 0.78 LMNA (0.38) LMNAPOLBCTSSCTSKAAK1
SCHEMBL17169209 0.78 LMNA (0.39) LMNAPOLBCTSSCTSKAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015156421-A1 DIHYDROTHIAZINE AND DIHYDROOXAZINE DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2015-10-15 WO disclosed