SCHEMBL1718102

SCHEMBL1718102

O=C(NCc1cccnc1)c1nn2c(C(F)(F)F)cc(-c3ccco3)nc2c1Cl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.65
ALDH1A1 P00352 13/20 0.58
HPGD P15428 6/20 0.58
NPSR1 Q6W5P4 4/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
MAPT P10636 6/20 0.54
CASP1 P29466 5/20 0.54
GAA P10253 2/20 0.54
ADORA3 P0DMS8 1/20 0.54
ADORA2A P29274 1/20 0.54
ADORA2B P29275 1/20 0.54
ADORA1 P30542 1/20 0.54
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
PKM P14618 2/20 0.51
NPC1 O15118 1/20 0.51
HTT P42858 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719162 0.91 KDM4E (0.70) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1719406 0.88 KDM4E (0.69) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1717864 0.86 ALDH1A1 (0.75) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1719980 0.85 ALDH1A1 (0.57) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1719624 0.84 ALDH1A1 (0.58) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1718948 0.84 ALDH1A1 (0.64) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL12239908 0.83 KDM4E (0.67) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1718997 0.82 ALDH1A1 (0.68) KDM4EALDH1A1HPGDCYP3A4CYP2C19
SCHEMBL1719199 0.82 ALDH1A1 (0.71) KDM4EALDH1A1HPGDNPSR1CYP1A2
SCHEMBL1719032 0.82 KDM4E (0.79) KDM4EALDH1A1HPGDNPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed