SCHEMBL1718948

SCHEMBL1718948

O=C(NCc1cccnc1)c1nn2c(C(F)(F)F)cc(-c3cccs3)nc2c1Cl

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.64
MAPT P10636 8/20 0.64
KDM4E B2RXH2 7/20 0.64
POLB P06746 3/20 0.64
KMT2A Q03164 4/20 0.62
MEN1 O00255 3/20 0.62
NPSR1 Q6W5P4 2/20 0.57
ESR1 P03372 1/20 0.57
BLM P54132 1/20 0.57
LMNA P02545 2/20 0.53
HPGD P15428 5/20 0.51
CASP1 P29466 3/20 0.51
CASP7 P55210 3/20 0.51
HSD17B10 Q99714 3/20 0.51
MYC P01106 1/20 0.50
MAX P61244 1/20 0.50
NPC1 O15118 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1718418 0.90 ALDH1A1 (0.70) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719114 0.88 KMT2A (0.66) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719980 0.85 ALDH1A1 (0.57) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719624 0.84 ALDH1A1 (0.58) ALDH1A1MAPTKDM4EPOLBNPSR1
SCHEMBL1718102 0.84 KDM4E (0.65) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719199 0.82 ALDH1A1 (0.71) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1718393 0.82 KMT2A (0.67) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719508 0.82 KMT2A (0.62) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719293 0.81 MAPT (0.65) ALDH1A1MAPTKDM4EPOLBKMT2A
SCHEMBL1719301 0.80 ALDH1A1 (0.76) ALDH1A1MAPTKDM4EPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed