SCHEMBL1718401

SCHEMBL1718401

O=C(Nc1ccccc1C(F)(F)F)c1cc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)n2n1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.72
KDM4E B2RXH2 4/20 0.66
ALDH1A1 P00352 2/20 0.66
SMN1; SMN2 Q16637 3/20 0.62
THRB P10828 4/20 0.61
HPGD P15428 4/20 0.60
MAPT P10636 3/20 0.59
HSD17B10 Q99714 2/20 0.59
RXFP1 Q9HBX9 3/20 0.57
TSHR P16473 1/20 0.56
RAB9A P51151 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1717969 0.92 TP53 (0.72) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1717962 0.91 TP53 (0.71) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1719086 0.89 TP53 (0.81) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1718728 0.89 TP53 (0.69) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1718632 0.87 THRB (0.75) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1719020 0.86 TP53 (0.85) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1718209 0.86 KDM4E (0.62) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1718976 0.85 THRB (0.77) TP53ALDH1A1SMN1; SMN2THRBHPGD
SCHEMBL1718532 0.83 THRB (0.84) TP53KDM4EALDH1A1SMN1; SMN2THRB
SCHEMBL1718195 0.83 MAPT (0.74) TP53KDM4EALDH1A1SMN1; SMN2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed