SCHEMBL1719086

SCHEMBL1719086

COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4ccccc4C(F)(F)F)cc3n2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.81
ALDH1A1 P00352 7/20 0.71
KDM4E B2RXH2 5/20 0.71
HPGD P15428 5/20 0.71
HSD17B10 Q99714 4/20 0.71
CASP1 P29466 3/20 0.71
CASP7 P55210 3/20 0.71
MAPT P10636 6/20 0.68
SMN1; SMN2 Q16637 2/20 0.68
TSHR P16473 2/20 0.65
USP2 O75604 1/20 0.65
ALOX15 P16050 1/20 0.65
THRB P10828 2/20 0.63
RXFP1 Q9HBX9 1/20 0.63
POLB P06746 1/20 0.62
CHRM4 P08173 1/20 0.62
GAA P10253 1/20 0.61
MEN1 O00255 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1718157 0.91 TP53 (0.81) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1718401 0.89 TP53 (0.72) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1717969 0.89 TP53 (0.72) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1717962 0.88 TP53 (0.71) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1718605 0.85 MAPT (0.73) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1718362 0.85 THRB (0.82) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1719103 0.84 TP53 (0.70) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1718263 0.84 MAPT (0.75) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL20467403 0.84 ALDH1A1 (0.77) TP53ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1718635 0.84 ALDH1A1 (0.75) TP53ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed