SCHEMBL1718407

SCHEMBL1718407

O=C(NCc1ccccc1)c1cc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2n1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.83
HPGD P15428 6/20 0.78
POLB P06746 4/20 0.78
HSD17B10 Q99714 3/20 0.78
CASP1 P29466 2/20 0.78
CASP7 P55210 2/20 0.78
LMNA P02545 1/20 0.78
BAP1 Q92560 1/20 0.78
THRB P10828 2/20 0.64
RXFP1 Q9HBX9 1/20 0.64
MAPT P10636 4/20 0.64
TP53 P04637 3/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
KDM4E B2RXH2 5/20 0.55
L3MBTL1 Q9Y468 2/20 0.54
USP2 O75604 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1718482 0.93 ALDH1A1 (0.80) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1718435 0.91 ALDH1A1 (1.00) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1719197 0.91 ALDH1A1 (0.78) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1718614 0.89 HPGD (0.74) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1717790 0.87 ALDH1A1 (1.00) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1719150 0.85 HPGD (0.63) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1719343 0.85 ALDH1A1 (0.68) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1718976 0.84 THRB (0.77) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1717957 0.84 TTR (0.70) ALDH1A1HPGDPOLBHSD17B10CASP1
SCHEMBL1718061 0.84 TP53 (0.67) ALDH1A1HPGDPOLBHSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed