SCHEMBL17184706

SCHEMBL17184706

COC(=O)c1ccc(C)c(Oc2ccc(Cl)c(F)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.52
ALDH1A1 P00352 5/20 0.44
HTR2A P28223 2/20 0.43
SLC6A4 P31645 2/20 0.43
KCNH2 Q12809 2/20 0.43
KMT2A Q03164 3/20 0.42
MAPT P10636 3/20 0.42
MEN1 O00255 1/20 0.42
CASP3 P42574 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
USP2 O75604 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
LMNA P02545 2/20 0.41
TDP1 Q9NUW8 1/20 0.40
GAA P10253 1/20 0.40
ICAM1 P05362 1/20 0.40
SELE P16581 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17184661 0.83 HTR2A (0.51) ALDH1A1HTR2ASLC6A4KCNH2KMT2A
SCHEMBL15968586 0.80 ALDH1A1 (0.58) NOTUMALDH1A1KMT2AMAPTMEN1
SCHEMBL29825107 0.80 ALDH1A1 (0.58) NOTUMALDH1A1KMT2AMAPTMEN1
SCHEMBL2671292 0.77 NOTUM (0.46) NOTUMALDH1A1KMT2AMAPTUSP2
SCHEMBL21363204 0.76 NOTUM (0.57) NOTUMALDH1A1KMT2AMAPTCASP3
SCHEMBL370483 0.76 USP2 (0.49) ALDH1A1KMT2AMAPTMEN1USP2
SCHEMBL26563554 0.74 CARM1 (0.50) NOTUMALDH1A1KMT2AMAPTMEN1
SCHEMBL16319599 0.74 SCN9A (0.52) NOTUMMAPTLMNAGAASCN9A
SCHEMBL22169879 0.74 KMT2A (0.59) NOTUMALDH1A1KMT2AMAPTUSP2
SCHEMBL17185227 0.73 ALDH1A1 (0.55) NOTUMALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161014-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed
WO-2015161011-A1 BENZAMIDE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed