SCHEMBL17185049

SCHEMBL17185049

NC(=O)c1cccc(C2CCOCC2)c1C1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.46
IKBKB O14920 1/20 0.42
CHUK O15111 1/20 0.42
PARP2 Q9UGN5 3/20 0.41
SIRT2 Q8IXJ6 1/20 0.39
HTR2C P28335 3/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
CDC7 O00311 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28325510 0.83 PARP1 (0.57) PARP1IKBKBCHUKPARP2SIRT2
SCHEMBL1006493 0.78 IKBKB (0.53) PARP1IKBKBCHUKPARP2SIRT2
SCHEMBL364173 0.78 ADRA1A (0.46) PARP1SIRT2CYP11B1CYP11B2
SCHEMBL31748898 0.77 CYP11B1 (0.43) PARP1PARP2CYP11B1CYP11B2AURKA
SCHEMBL28853765 0.77 PARP1 (0.52) PARP1IKBKBCHUKPARP2HTR2C
SCHEMBL1004217 0.77 MEN1 (0.49) PARP1PARP2
Hydrochloric Acid SCHEMBL28243995 0.77 HTR2C (0.53) PARP1IKBKBCHUKPARP2SIRT2
SCHEMBL3809365 0.76 PARP1 (0.51) PARP1IKBKBCHUKPARP2HTR2C
SCHEMBL3809376 0.76 HTR2C (0.59) PARP1IKBKBCHUKPARP2HTR2C
SCHEMBL20822489 0.76 CYP11B1 (0.42) PARP1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161011-A1 BENZAMIDE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed