SCHEMBL1718653

SCHEMBL1718653

O=C(c1cc2nc(-c3cccs3)cc(C(F)(F)F)n2n1)N1CCN(C(=O)c2ccco2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 15/20 0.70
ALDH1A1 P00352 13/20 0.70
HPGD P15428 11/20 0.70
HSD17B10 Q99714 8/20 0.70
CASP1 P29466 6/20 0.70
CASP7 P55210 6/20 0.70
KLK7 P49862 1/20 0.65
HTT P42858 3/20 0.64
APOBEC3A P31941 1/20 0.64
MAPT P10636 8/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
LMNA P02545 5/20 0.62
USP2 O75604 4/20 0.62
ALOX15 P16050 2/20 0.62
RECQL P46063 1/20 0.62
NPSR1 Q6W5P4 5/20 0.60
GAA P10253 3/20 0.60
TSHR P16473 2/20 0.60
MAPK1 P28482 2/20 0.57
RXFP1 Q9HBX9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4197490 0.87 KDM4E (0.74) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL1718960 0.86 KDM4E (0.72) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL1718295 0.86 KDM4E (0.72) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL1718993 0.85 KDM4E (0.71) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL4211222 0.84 ALDH1A1 (0.69) KDM4EALDH1A1HPGDHSD17B10KLK7
SCHEMBL1719204 0.82 ALDH1A1 (0.70) KDM4EALDH1A1HPGDHSD17B10KLK7
SCHEMBL4210939 0.82 KDM4E (0.66) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL4207198 0.81 HPGD (0.76) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL4204177 0.80 KDM4E (0.70) KDM4EALDH1A1HPGDHSD17B10CASP1
SCHEMBL4200688 0.79 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed