SCHEMBL1719352

SCHEMBL1719352

COc1cc2ncnc(Oc3ccc(CC(=O)Nc4nc(C)c(C)s4)cc3)c2cc1OC

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 11/20 0.65
FLT3 P36888 9/20 0.65
FLT4 P35916 9/20 0.65
CSF1R P07333 5/20 0.65
KDR P35968 8/20 0.60
CYP2C9 P11712 1/20 0.60
PDGFRA P16234 1/20 0.55
ROCK2 O75116 1/20 0.53
MET P08581 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1099153 0.94 PDGFRB (0.59) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4185538 0.89 PDGFRB (0.51) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1099216 0.86 PDGFRB (0.66) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1097598 0.86 PDGFRB (0.65) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4669695 0.85 KDR (0.74) PDGFRBFLT4CSF1RKDRPDGFRA
SCHEMBL1099731 0.82 KDR (0.54) PDGFRBFLT4CSF1RKDRPDGFRA
SCHEMBL1099936 0.82 KDR (0.54) PDGFRBFLT4CSF1RKDRPDGFRA
SCHEMBL4371744 0.82 MET (0.77) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL20788539 0.82 KMT2A (0.64) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1098052 0.81 PDGFRB (0.60) PDGFRBFLT3FLT4CSF1RKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802591-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2012-01-11 EP claimed