SCHEMBL1719647

SCHEMBL1719647

O=c1[nH]c2onc(C3CCNCC3)c2c2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.39
HTR2C P28335 3/20 0.38
HTR2A P28223 1/20 0.38
KCNH2 Q12809 1/20 0.38
GABRA1 P14867 3/20 0.38
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
SLC18A3 Q16572 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
ADRB2 P07550 1/20 0.35
KHK P50053 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1719910 0.99 PARP1 (0.38) PARP1HTR2CHTR2AKCNH2GABRA1
SCHEMBL1720278 0.84 PARP1 (0.49) PARP1HTR2A
SCHEMBL1719871 0.81 PARP1 (0.63) PARP1HTR2A
SCHEMBL1720062 0.77 PARP1 (0.41) PARP1
SCHEMBL1720663 0.76 ALDH1A1 (0.47) PARP1
SCHEMBL12845934 0.73 ATM (0.45) PARP1HTR2CHTR2AKCNH2GABRA1
SCHEMBL1719884 0.72 PARP1 (0.71) PARP1HTR2CHTR2AKCNH2KHK
SCHEMBL1720694 0.71 PARP1 (0.41) PARP1
SCHEMBL373467 0.71 BCHE (0.44) HTR2CHTR2ASLC18A3SIGMAR1ADRB2
Hydrochloric Acid SCHEMBL1719792 0.71 PARP1 (0.70) PARP1HTR2CHTR2AKCNH2KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP claimed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed