SCHEMBL373467

SCHEMBL373467

c1ccc2c(C3CCNCC3)noc2c1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
SLC18A3 Q16572 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HTR1A P08908 8/20 0.42
DRD2 P14416 8/20 0.42
HTR2A P28223 8/20 0.42
MAPK14 Q16539 1/20 0.42
ADRB2 P07550 1/20 0.41
HTR2C P28335 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5995383 0.98 BCHE (0.43) BCHEACHESLC18A3SIGMAR1HTR1A
Hydrochloric Acid SCHEMBL1545403 0.98 BCHE (0.43) BCHEACHESLC18A3SIGMAR1HTR1A
SCHEMBL9377809 0.90 HTR1A (0.39) BCHEACHEHTR1ADRD2HTR2A
SCHEMBL7726651 0.88 ACHE (0.55) ACHEDRD2HTR2AHTR2C
SCHEMBL23175425 0.88 DRD2 (0.46) HTR1ADRD2HTR2A
SCHEMBL12026856 0.83 HIF1A (0.49) ACHEHTR1ADRD2HTR2A
SCHEMBL795369 0.81 HTR2A (0.44) HTR1ADRD2HTR2AHTR2C
SCHEMBL3263185 0.81 DRD2 (0.44) HTR1ADRD2HTR2A
SCHEMBL7966226 0.80 DRD2 (0.39) HTR1ADRD2HTR2A
SCHEMBL7966228 0.80 DRD2 (0.39) HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 166 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102796090-B Method for preparing iloperidone TIANJIN HUAJIN PHARMACEUTICAL CO LTD 2015-03-25 CN claimed
CN-102070626-A Novel method for preparing iloperidone HAINAN KANGHONG PHARMACEUTICAL R & D CO LTD 2011-05-25 CN claimed
EP-0760811-A1 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H 3? (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-03-12 EP claimed
US-5385916-A 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents PFIZER INC. (US) 1995-01-31 US claimed
EP-0557289-B1 4-(1,2-BENZISOXAZOLYL)PIPERIDINE ANTIPSYCHOTIC AGENTS PFIZER (US) 1994-12-28 EP claimed
US-5276040-A 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents PFIZER INC. (US) 1994-01-04 US claimed
US-5147881-A 4-(1,2-BENZISOXAZOLYL)PIPERIDINE ANTIPSYCHOTIC AGENTS PFIZER INC (US) 1992-09-15 US claimed
WO-1992008718-A1 4-(1,2-BENZISOXAZOLYL)PIPERIDINE ANTIPSYCHOTIC AGENTS PFIZER INC. (US) 1992-05-29 WO claimed
EP-0080104-B1 3-(4-PIPERIDYL)-1,2-BENZISOXAZOLES, PROCESS FOR THE PREPARATION THEREOF, AND A PHARMACEUTICAL COMPOSITION COMPRISING THE SAME HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-12-14 EP claimed
EP-0080104-A2 3-(4-Piperidyl)-1,2-benzisoxazoles, process for the preparation thereof, and a pharmaceutical composition comprising the same HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-06-01 EP claimed
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US claimed
JP-10059967-A None JP disclosed
JP-58090582-A None JP disclosed
US-20260078115-A1 ALIPHATIC ACID AMIDE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2026-03-19 US disclosed
US-12503463-B2 Aliphatic acid amide derivative Sumitomo Pharma Co., Ltd. (JP) 2025-12-23 US disclosed
JP-S5890582-A 3-(4-PIPERIDYL)-1,2-BENZISOXAZOLE COMPOUND HOECHST ROUSSEL PHARMA 1983-05-30 JP disclosed
EP-0079564-A1 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles, a process for the preparation thereof, a pharmaceutical composition comprising the same, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-05-25 EP disclosed
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US disclosed
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US disclosed
US-4352811-A NEUROLEPTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1982-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503463-B2 Aliphatic acid amide derivative HTR2A, HTR1A, HTR7 BCHE 3307/4885ACHE 1920/4885SLC18A3 593/4885
US-20260078115-A1 ALIPHATIC ACID AMIDE DERIVATIVE HTR1D, HTR1A, HTR7 BCHE 2651/4885ACHE 2428/4885SLC18A3 912/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.