SCHEMBL17199895

SCHEMBL17199895

O=C(NCc1ccc(OCc2cccc(C(F)(F)F)c2)cc1)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)s1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.54
MMP1 P03956 2/20 0.51
ADAM17 P78536 2/20 0.51
MMP8 P22894 1/20 0.46
MMP12 P39900 1/20 0.46
MMP13 P45452 1/20 0.46
PDGFRA P16234 1/20 0.46
S1PR1 P21453 1/20 0.46
S1PR5 Q9H228 1/20 0.46
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.43
AADAT Q8N5Z0 1/20 0.42
FFAR1 O14842 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
FKBP1A P62942 1/20 0.42
NR4A2 P43354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17136569 0.94 TRPA1 (0.52) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199902 0.93 TRPA1 (0.58) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136492 0.93 TRPA1 (0.53) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199898 0.91 TRPA1 (0.61) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136474 0.91 TRPA1 (0.61) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199887 0.89 TRPA1 (0.56) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136454 0.89 TRPA1 (0.55) TRPA1MMP8MMP12MMP13HCRTR1
SCHEMBL17199901 0.88 TRPA1 (0.53) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136565 0.87 TRPA1 (0.54) TRPA1MMP8MMP12MMP13HCRTR1
SCHEMBL17136379 0.87 TRPA1 (0.52) TRPA1MMP8MMP12MMP13HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2937335-A1 HETEROCYCLIC AMIDE DERIVATIVE, AND MEDICINE CONTAINING SAME Ajinomoto Co., Inc. (JP) 2015-10-28 EP disclosed