SCHEMBL17199898

SCHEMBL17199898

O=C(NCc1ccc(OCc2ccc(C(F)(F)F)cc2)cc1)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)s1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 6/20 0.61
MMP1 P03956 1/20 0.49
ADAM17 P78536 1/20 0.49
MMP8 P22894 1/20 0.49
MMP12 P39900 1/20 0.49
MMP13 P45452 1/20 0.49
ALDH1A1 P00352 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
HDAC1 Q13547 3/20 0.44
HDAC2 Q92769 3/20 0.44
HDAC3 O15379 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17136474 1.00 TRPA1 (0.61) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199918 0.93 TRPA1 (0.64) TRPA1MMP8MMP12MMP13ALDH1A1
SCHEMBL17199902 0.92 TRPA1 (0.58) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136379 0.92 TRPA1 (0.52) TRPA1MMP8MMP12MMP13ALDH1A1
SCHEMBL17199895 0.91 TRPA1 (0.54) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199887 0.91 TRPA1 (0.56) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136418 0.91 MMP8 (0.54) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136513 0.91 MMP8 (0.53) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17136492 0.91 TRPA1 (0.53) TRPA1MMP1ADAM17MMP8MMP12
SCHEMBL17199908 0.90 TRPA1 (0.60) TRPA1MMP1ADAM17MMP8MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2937335-A1 HETEROCYCLIC AMIDE DERIVATIVE, AND MEDICINE CONTAINING SAME Ajinomoto Co., Inc. (JP) 2015-10-28 EP disclosed