SCHEMBL17201973

SCHEMBL17201973

Nc1ccnc(-c2cnc(N3CCC(F)(F)CC3)nc2N)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 13/20 0.47
KCNK2 O95069 1/20 0.36
SCN2A Q99250 1/20 0.36
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
TRPV3 Q8NET8 1/20 0.35
PRKCA P17252 1/20 0.35
PRKCQ Q04759 1/20 0.35
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
ROCK2 O75116 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17201969 0.87 PTPN11 (0.39) PTPN11KCNK2SCN2AROCK2
SCHEMBL17202011 0.86 GSK3A (0.37) PTPN11GSK3AGSK3BTRPV3PIK3CA
SCHEMBL22119525 0.81 OGA (0.44) PTPN11GSK3AGSK3BTRPV3PIK3CA
SCHEMBL17610067 0.77 DYRK1A (0.41) PTPN11KCNK2SCN2A
SCHEMBL17201967 0.77 PTPN11 (0.38) PTPN11PIK3CAMTOR
SCHEMBL26975257 0.73 PTPN11 (0.46) PTPN11TRPV3PRKCAPRKCQ
SCHEMBL17201976 0.72 MAP3K12 (0.34) PIK3CAMTORROCK2
SCHEMBL17201937 0.71 DYRK1A (0.45) PIK3CAMTOR
SCHEMBL17202180 0.71 TRPA1 (0.40) PTPN11PIK3CAMTOR
SCHEMBL17201952 0.70 DYRK1A (0.42) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134410-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Hydra Biosciences, Inc. (US) 2017-03-01 EP disclosed
WO-2015164643-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2015-10-29 WO disclosed