SCHEMBL17202027

SCHEMBL17202027

CC1CCCN1c1ncc(-c2nccc(N)n2)cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 3/20 0.47
DYRK1A Q13627 1/20 0.45
PIM1 P11309 2/20 0.40
PIM3 Q86V86 2/20 0.40
PIM2 Q9P1W9 2/20 0.40
SMPD3 Q9NY59 1/20 0.40
PBRM1 Q86U86 5/20 0.40
LRRK2 Q5S007 1/20 0.38
SMARCA2 P51531 4/20 0.38
SMARCA4 P51532 3/20 0.38
NR1I2 O75469 2/20 0.38
NR1H2 P55055 1/20 0.38
PIK3CA P42336 4/20 0.37
MTOR P42345 4/20 0.37
PIK3R1 P27986 2/20 0.37
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18539056 1.00 MAP3K12 (0.47) MAP3K12DYRK1APIM1PIM3PIM2
SCHEMBL17210369 1.00 MAP3K12 (0.47) MAP3K12DYRK1APIM1PIM3PIM2
SCHEMBL17210359 0.96 MAP3K12 (0.43) MAP3K12DYRK1APIM1PIM3PIM2
SCHEMBL17201937 0.86 DYRK1A (0.45) MAP3K12DYRK1APIM1PIM3PIM2
SCHEMBL17201952 0.83 DYRK1A (0.42) MAP3K12DYRK1APIM1PIM3PIM2
SCHEMBL24942475 0.82 DYRK1A (0.51) MAP3K12DYRK1ASMPD3PBRM1LRRK2
SCHEMBL24942471 0.82 DYRK1A (0.51) MAP3K12DYRK1ASMPD3PBRM1LRRK2
SCHEMBL17210340 0.81 TRPA1 (0.49) PIK3CAMTOR
SCHEMBL17202009 0.81 TRPA1 (0.49) PIK3CAMTOR
SCHEMBL17205369 0.81 TRPA1 (0.49) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134410-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Hydra Biosciences, Inc. (US) 2017-03-01 EP disclosed
WO-2015164643-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2015-10-29 WO disclosed