SCHEMBL17215007

SCHEMBL17215007

COc1ccc2cc(-c3ccc(I)o3)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.51
HSD17B2 P37059 2/20 0.51
GSTP1 P09211 1/20 0.49
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
ABCB1 P08183 1/20 0.45
CYP11B1 P15538 4/20 0.45
CYP11B2 P19099 4/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
APP P05067 3/20 0.44
CYP2A6 P11509 2/20 0.44
PDE4A P27815 1/20 0.43
CYP17A1 P05093 1/20 0.43
CYP19A1 P11511 1/20 0.43
MAOB P27338 1/20 0.43
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18551784 0.81 GSK3B (0.56) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL18539942 0.79 HSD17B1 (0.50) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL11723032 0.75 HSD17B1 (0.83) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL12051687 0.75 HSD17B1 (0.83) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL3020390 0.72 HSD17B1 (0.76) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL22106285 0.72 HSD17B1 (0.76) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL14041533 0.72 HSD17B1 (0.76) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL6579774 0.71 APP (0.60) NPC1RAB9ACYP1A2CYP3A4APP
SCHEMBL29447161 0.71 CYP1A2 (0.79) HSD17B1HSD17B2GSTP1NPC1RAB9A
SCHEMBL443070 0.71 CYP1A2 (0.79) HSD17B1HSD17B2GSTP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015164411-A9 SMALL MOLECULE INHIBITORS OF G PROTEIN COUPLED RECEPTOR 6 KINASE POLYPEPTIDES MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2016-05-26 WO disclosed
WO-2015164411-A2 SMALL MOLECULE INHIBITORS OF G PROTEIN COUPLED RECEPTOR 6 KINASES POLYPEPTIDES MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2015-10-29 WO disclosed