SCHEMBL17220116

SCHEMBL17220116

CC(C)N(c1ccccc1)c1nc(N)nc(C(N)=NO)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
TP53 P04637 1/20 0.45
ALOX15 P16050 1/20 0.45
DHFR P00374 4/20 0.45
MAPT P10636 4/20 0.37
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
JAK2 O60674 1/20 0.33
ALDH1A1 P00352 3/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
PRNP P04156 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HTT P42858 2/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL795288 0.82 TSHR (0.48) TSHRTP53ALOX15DHFRMAPT
SCHEMBL796712 0.82 TSHR (0.48) TSHRTP53ALOX15DHFRMAPT
SCHEMBL8608925 0.79 DHFR (0.45) TSHRTP53DHFRMAPTLMNA
SCHEMBL17220453 0.79 TSHR (0.48) TSHRTP53ALOX15DHFRMAPT
SCHEMBL17220115 0.78 DHFR (0.44) TSHRDHFRMAPTLMNASMN1; SMN2
SCHEMBL7700052 0.75 DHFR (0.51) TSHRDHFRMAPTLMNASMN1; SMN2
SCHEMBL795662 0.74 TSHR (0.41) TSHRTP53ALOX15DHFRMAPT
SCHEMBL17220137 0.74 TSHR (0.41) TSHRTP53ALOX15DHFRMAPT
SCHEMBL17220070 0.74 SMN1; SMN2 (0.45) TSHRTP53ALOX15DHFRMAPT
SCHEMBL17220364 0.73 TSHR (0.45) TSHRTP53ALOX15DHFRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616465-B1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2015-11-04 EP disclosed