SCHEMBL17220137

SCHEMBL17220137

COCCN(c1ccccc1)c1nc(N)nc(/C(N)=N/O)n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPT P10636 3/20 0.36
DHFR P00374 6/20 0.35
NPC1 O15118 1/20 0.33
JAK2 O60674 1/20 0.33
RAB9A P51151 1/20 0.33
KCNA3 P22001 1/20 0.32
KCNA5 P22460 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CRHBP P24387 1/20 0.30
CRHR2 Q13324 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL795662 1.00 TSHR (0.41) TSHRTP53ALOX15MAPTDHFR
SCHEMBL17220453 0.84 TSHR (0.48) TSHRTP53ALOX15MAPTDHFR
SCHEMBL795663 0.81 MAPT (0.35) MAPTDHFRNPC1JAK2RAB9A
SCHEMBL17220160 0.78 DHFR (0.41) TSHRMAPTDHFRNPC1JAK2
SCHEMBL17220364 0.78 TSHR (0.45) TSHRTP53ALOX15MAPTDHFR
SCHEMBL795288 0.77 TSHR (0.48) TSHRTP53ALOX15MAPTDHFR
SCHEMBL796712 0.77 TSHR (0.48) TSHRTP53ALOX15MAPTDHFR
SCHEMBL796138 0.75 MAPT (0.59) TSHRMAPTDHFRNPC1JAK2
SCHEMBL17220116 0.74 TSHR (0.45) TSHRTP53ALOX15MAPTDHFR
SCHEMBL17220376 0.72 MTNR1A (0.39) TSHRTP53ALOX15DHFRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616465-B1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2015-11-04 EP disclosed