SCHEMBL172250

SCHEMBL172250

CCC(CN(C)CCC(C)C)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.50
HTR2A P28223 4/20 0.43
HRH1 P35367 4/20 0.43
AOC3 Q16853 4/20 0.41
TDP1 Q9NUW8 1/20 0.40
SIGMAR1 Q99720 2/20 0.39
LMNA P02545 2/20 0.37
OPRM1 P35372 2/20 0.36
SLC22A1 O15245 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
CYP1A2 P05177 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2D6 P10635 1/20 0.35
CHRM1 P11229 1/20 0.35
TSHR P16473 1/20 0.35
ADRA2B P18089 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096616 0.80 AOC3 (0.58) HTR2AHRH1AOC3TDP1TAAR1
SCHEMBL13948770 0.79 CCR5 (0.47) CCR5HTR2AHRH1TDP1SIGMAR1
SCHEMBL21739939 0.77 HTR2A (0.61) CCR5HTR2AHRH1AOC3TDP1
SCHEMBL21739938 0.77 HTR2A (0.61) CCR5HTR2AHRH1AOC3TDP1
SCHEMBL3428926 0.77 HTR2A (0.61) CCR5HTR2AHRH1AOC3TDP1
SCHEMBL13995351 0.77 AOC3 (0.59) HTR2AHRH1AOC3LMNATAAR1
SCHEMBL3068671 0.77 HRH1 (0.62) HTR2AHRH1AOC3TDP1SIGMAR1
SCHEMBL23138901 0.74 HTR2A (0.64) CCR5HTR2AHRH1TDP1SIGMAR1
SCHEMBL22426629 0.74 CCR5 (0.44) CCR5HTR2AHRH1AOC3TDP1
SCHEMBL12300267 0.74 HTR2A (0.64) CCR5HTR2AHRH1TDP1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed