SCHEMBL17226352

SCHEMBL17226352

CC(C)Nc1cc(C#CC(C)(C)C)sc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.38
CYP2E1 P05181 1/20 0.36
HCAR3 P49019 1/20 0.35
ALDH1A1 P00352 1/20 0.32
PTPRF P10586 1/20 0.30
PTPN1 P18031 1/20 0.30
PTPRA P18433 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14645197 0.86 RAF1 (0.35)
SCHEMBL1082972 0.85 NR1I2 (0.37) NR1I2CYP2E1HCAR3ALDH1A1
SCHEMBL17226353 0.84 NR1I2 (0.38) NR1I2CYP2E1HCAR3PTPRFPTPN1
SCHEMBL15015340 0.78 RAB9A (0.42) NR1I2CYP2E1HCAR3ALDH1A1PTPN1
SCHEMBL15015299 0.77 NR1I2 (0.33) NR1I2CYP2E1
SCHEMBL16661952 0.77 NR1I2 (0.41) NR1I2CYP2E1L3MBTL1
SCHEMBL15130828 0.76 ALDH1A1 (0.36) ALDH1A1
SCHEMBL19364937 0.76 NR1I2 (0.40) NR1I2CYP2E1ALDH1A1L3MBTL1
SCHEMBL432666 0.75 NR1I2 (0.39) NR1I2CYP2E1L3MBTL1
SCHEMBL12949396 0.75 NR1I2 (0.39) NR1I2CYP2E1PTPN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403860-B1 PHOSPHOTHIOPHENE AND PHOSPHOTHIAZOLE AS HCV POLYMERASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2015-11-04 EP disclosed