SCHEMBL17226505

SCHEMBL17226505

C=C(C)CN1CCC(CCN2CCN(c3cccc(CC(C)C)c3)CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.44
DRD2 P14416 6/20 0.43
DRD3 P35462 6/20 0.43
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SIGMAR1 Q99720 2/20 0.41
ADRB1 P08588 1/20 0.39
HRH1 P35367 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
OPRM1 P35372 1/20 0.39
HTR1A P08908 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3845038 0.90 DRD2 (0.47) VCPDRD2DRD3SLC6A2SLC6A4
SCHEMBL14346806 0.85 NOTUM (0.45) VCPDRD2DRD3SLC6A2SLC6A4
SCHEMBL3853616 0.82 DRD2 (0.48) VCPDRD2DRD3SLC6A2SLC6A4
SCHEMBL4496072 0.79 GPR119 (0.54) VCPDRD2DRD3
SCHEMBL3853660 0.78 DRD2 (0.50) DRD2DRD3SLC6A2SLC6A4
SCHEMBL3853868 0.78 DRD2 (0.50) DRD2DRD3SLC6A2SLC6A4
SCHEMBL3845208 0.76 DRD2 (0.48) DRD2DRD3SLC6A2SLC6A4SIGMAR1
SCHEMBL3843937 0.76 DRD2 (0.53) DRD2DRD3SLC6A2SLC6A4SIGMAR1
SCHEMBL14346795 0.76 GFER (0.47) DRD2DRD3SLC6A2SLC6A4
SCHEMBL3847168 0.76 DRD2 (0.47) DRD2DRD3SLC6A2SLC6A4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038268-B1 CARBONYLATED (AZA)CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2015-11-04 EP disclosed