SCHEMBL17227458

SCHEMBL17227458

COC(=O)N1CC2(CCN(C(=O)Cc3ccc(OC)cc3)CC2)C1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.66
MAPT P10636 2/20 0.60
GHSR Q92847 4/20 0.57
CYP3A4 P08684 4/20 0.57
CYP2C19 P33261 2/20 0.57
CYP2C9 P11712 1/20 0.57
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 2/20 0.54
TSHR P16473 1/20 0.54
GFER P55789 1/20 0.53
CHRM2 P08172 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
HPGD P15428 3/20 0.51
ALDH1A1 P00352 2/20 0.51
KMT2A Q03164 1/20 0.51
HSD17B10 Q99714 1/20 0.51
GAA P10253 1/20 0.50
USP2 O75604 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2441294 0.89 SMN1; SMN2 (0.68) SMN1; SMN2MAPTGHSRGFERCHRM2
SCHEMBL2445002 0.88 SMN1; SMN2 (0.60) SMN1; SMN2MAPTGHSRCYP3A4GFER
SCHEMBL12328016 0.86 GHSR (0.59) SMN1; SMN2MAPTGHSRCYP3A4GFER
SCHEMBL12299405 0.83 SMN1; SMN2 (0.71) SMN1; SMN2MAPTGHSRGFERCHRM2
SCHEMBL17227462 0.82 GHSR (0.61) GHSRCYP3A4CYP2C19CYP2C9CHRM2
Hydrochloric Acid SCHEMBL2431655 0.82 SMN1; SMN2 (0.69) SMN1; SMN2MAPTGHSRGFERCHRM2
SCHEMBL2236750 0.77 SMN1; SMN2 (0.84) SMN1; SMN2MAPTGFERL3MBTL1HPGD
SCHEMBL9321597 0.76 MAPT (1.00) SMN1; SMN2MAPTGFERL3MBTL1HPGD
SCHEMBL92507 0.76 SMN1; SMN2 (0.82) SMN1; SMN2MAPTGFERL3MBTL1HPGD
SCHEMBL26099620 0.75 SMN1; SMN2 (0.55) SMN1; SMN2MAPTCYP3A4CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547679-B1 2,3 DIHYDRO-1H-INDEN-1-YL-2,7-DIAZASPIRO[3.6]NONANE DERIVATIVES AND THEIR USE AS ANTAGONISTS OR INVERSE AGONISTS OF THE GHRELIN RECEPTOR PFIZER (US) 2015-11-04 EP disclosed