SCHEMBL17227588

SCHEMBL17227588

COC(=O)c1sc(CC(C)C)cc1CBr

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.42
ALDH1A1 P00352 3/20 0.36
MAPT P10636 5/20 0.36
KMT2A Q03164 3/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
KDM4E B2RXH2 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 2/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
IKBKB O14920 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
GSK3B P49841 1/20 0.34
FEN1 P39748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14390861 0.78 RAF1 (0.43) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL2729001 0.78 GSK3B (0.43) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL21152318 0.76 IKBKB (0.42) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL13545972 0.76 RAF1 (0.39) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL161941 0.74 L3MBTL1 (0.60) RAF1MAPTL3MBTL1PKM
SCHEMBL1979077 0.73 RAF1 (0.51) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL12523234 0.73 RAF1 (0.51) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL24212419 0.73 L3MBTL1 (0.46) RAF1MAPTKMT2ATSHRHSD17B10
SCHEMBL13545968 0.72 ALDH1A1 (0.40) RAF1ALDH1A1MAPTKMT2ATSHR
SCHEMBL12272546 0.71 RAF1 (0.52) RAF1ALDH1A1MAPTKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611790-B1 PYRIDINONES/PYRAZINONES, METHOD OF MAKING, AND METHOD OF USE THEREOF GILEAD CONNECTICUT INC (US) 2015-11-04 EP disclosed