Floxuridine

Floxuridine

SCHEMBL17229

O=c1[nH]c(=O)n([C@@H]2CC(O)[C@H](CO)O2)cc1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TYMS

The experimentally established mechanism targets of Floxuridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 1.00
SMN1; SMN2 Q16637 2/20 1.00
TK1 P04183 3/20 0.73
ALOX12 P18054 1/20 0.72
ADRA1A P35348 1/20 0.72
TK2 O00142 1/20 0.67
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
TSHR P16473 1/20 0.66
BLM P54132 1/20 0.66
PMP22 Q01453 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Floxuridine SCHEMBL18561102 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL6270910 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL9155703 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL13674187 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL18573179 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL4939702 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL11564431 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL2050487 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL11563300 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A
Floxuridine SCHEMBL18597573 1.00 LMNA (1.00) LMNASMN1; SMN2TK1ALOX12ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6036 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137686-A1 SOLID PHARMACEUTICAL FORMULATION OF PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS SHANGHAI INC (CN) 2026-05-21 US claimed
US-20260137685-A1 SOLID PHARMACEUTICAL FORMULATION OF PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS SHANGHAI INC (CN) 2026-05-21 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-4711364-A1 FUSED PYRROLE RING OR FUSED PYRIDINE RING COMPOUND Pharmaengine, Inc. (TW) 2026-03-18 EP claimed
EP-4701737-A2 MTA-COOPERATIVE PRMT5 INHIBITOR Pharmaengine, Inc. (TW) 2026-03-04 EP claimed
US-12544378-B2 Solid pharmaceutical formulation of PARP inhibitors and use thereof Impact Therapeutics (Shanghai), Inc (CN) 2026-02-10 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4673448-A1 SUBSTITUTED NITROGEN-CONTAINING TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND THE USE THEREOF Impact Therapeutics (Shanghai), Inc. (CN) 2026-01-07 EP claimed
US-12492197-B2 3,5-disubstituted pyrazole compounds as kinase inhibitors and uses thereof Impact Therapeutics (Shanghai), Inc (CN) 2025-12-09 US claimed
US-12479848-B2 Substituted fused heteroaromatic bicyclic compounds as kinase inhibitors and the use thereof Impact Therapeutics (Shanghai), Inc (CN) 2025-11-25 US claimed
US-4599404-A BENOYLATION FUNAI PHARMACEUTICAL IND., LTD. (JP) 1986-07-08 US claimed
EP-0160079-A4 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION. GREER SHELDON B 1986-05-14 EP claimed
EP-0180188-A2 A composition for increasing the anti-cancer activity of an anti-cancer compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-05-07 EP claimed
EP-0160079-A1 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION. GREER SHELDON B 1985-11-06 EP claimed
EP-0151189-A1 ANTINEOPLASTIC AGENT TEIJIN LIMITED (JP) 1985-08-14 EP claimed
EP-0081386-B1 5-FLUORO-2'-DEOXYURIDINE DERIVATIVES AND A PROCESS FOR THE PREPARATION THEREOF TEIJIN LIMITED (JP) 1985-05-29 EP claimed
WO-1985001871-A1 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION GREER SHELDON B 1985-05-09 WO claimed
EP-0081386-A1 5-Fluoro-2'-deoxyuridine derivatives and a process for the preparation thereof TEIJIN LIMITED (JP) 1983-06-15 EP claimed
EP-0009882-B1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVES, A PROCESS FOR PRODUCING THE SAME AND ANTITUMOR AGENTS COMPRISING THE SAME FUNAI PHARMACEUTICAL IND., LTD. (JP) 1982-03-03 EP claimed
EP-0009882-A1 2'-Deoxy-5-fluorouridine derivatives, a process for producing the same and antitumor agents comprising the same FUNAI PHARMACEUTICAL IND., LTD. (JP) 1980-04-16 EP claimed