SCHEMBL17233302

SCHEMBL17233302

O=C(/C=C/c1cccnc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 9/20 1.00
CYP1A2 P05177 9/20 1.00
CYP1B1 Q16678 9/20 1.00
RAB9A P51151 4/20 0.74
MAPT P10636 2/20 0.74
KMT2A Q03164 1/20 0.74
PFKFB3 Q16875 1/20 0.73
CYP3A4 P08684 5/20 0.68
CYP2D6 P10635 5/20 0.68
NPC1 O15118 3/20 0.67
NTSR1 P30989 1/20 0.63
USP2 O75604 1/20 0.60
KDM4E B2RXH2 2/20 0.59
JUN P05412 1/20 0.59
NFKB1 P19838 1/20 0.59
MAPK1 P28482 1/20 0.59
GPR55 Q9Y2T6 1/20 0.59
P4HB P07237 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979409 0.91 CYP1B1 (0.83) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL7368933 0.91 CYP1B1 (0.83) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL13479662 0.91 RAB9A (0.88) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL29600034 0.85 RAB9A (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL5646960 0.85 RAB9A (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL1604140 0.85 RAB9A (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL29458617 0.84 PFKFB3 (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL196640 0.84 PFKFB3 (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL196639 0.84 PFKFB3 (1.00) CYP1A1CYP1A2CYP1B1RAB9AMAPT
SCHEMBL979407 0.84 CYP1B1 (0.78) CYP1A1CYP1A2CYP1B1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015166043-A1 COMPOUNDS DE MONTFORT UNIVERSITY (GB) 2015-11-05 WO disclosed