SCHEMBL17242599

SCHEMBL17242599

CC(O)Cn1c(=O)[nH]c(=O)c2ccccc21

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.49
BACE1 P56817 2/20 0.45
DAO P14920 1/20 0.44
AGER Q15109 1/20 0.43
IDO1 P14902 1/20 0.43
PARP2 Q9UGN5 3/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PER2 O15055 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6027770 0.88 SMN1; SMN2 (0.53) PARP1DAOPARP2ALDH1A1KDM4E
SCHEMBL30704833 0.88 SMN1; SMN2 (0.53) PARP1DAOPARP2ALDH1A1KDM4E
SCHEMBL6300121 0.85 PARP1 (0.46) PARP1DAOPARP2ALDH1A1
SCHEMBL10834234 0.81 MEN1 (0.63) DAOIDO1ALDH1A1
SCHEMBL6027805 0.79 CYP1A2 (0.64) PARP1DAOALDH1A1KDM4E
SCHEMBL30145436 0.78 BACE1 (0.70) BACE1AGERALDH1A1KDM4EPER2
SCHEMBL11788371 0.78 BACE1 (0.70) BACE1AGERALDH1A1KDM4EPER2
SCHEMBL6800624 0.78 DAO (0.43) PARP1BACE1DAOIDO1
SCHEMBL11983439 0.77 PARP1 (0.56) PARP1DAOPARP2KDM4E
SCHEMBL6295245 0.77 PARP1 (0.53) PARP1DAOPARP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3140301-A1 PHARMACOLOGICALLY ACTIVE QUINAZOLINEDIONE DERIVATIVES Orion Corporation (FI) 2017-03-15 EP claimed
WO-2015169999-A1 PHARMACOLOGICALLY ACTIVE QUINAZOLINEDIONE DERIVATIVES ORION CORPORATION (FI) 2015-11-12 WO claimed