SCHEMBL6300121

SCHEMBL6300121

C[C@@H](S)Cn1c(=O)[nH]c(=O)c2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.46
DAO P14920 1/20 0.44
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
PARP2 Q9UGN5 5/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30704833 0.88 SMN1; SMN2 (0.53) PARP1DAOCYP1A2PARP2ALDH1A1
SCHEMBL6027770 0.88 SMN1; SMN2 (0.53) PARP1DAOCYP1A2PARP2ALDH1A1
SCHEMBL6295245 0.85 PARP1 (0.53) PARP1DAOMEN1CYP1A2KMT2A
SCHEMBL17242599 0.85 PARP1 (0.49) PARP1DAOPARP2ALDH1A1
SCHEMBL6800624 0.84 DAO (0.43) PARP1DAOMEN1CYP1A2KMT2A
SCHEMBL6027805 0.79 CYP1A2 (0.64) PARP1DAOMEN1CYP1A2KMT2A
SCHEMBL6294349 0.76 PARP1 (0.52) PARP1DAOCYP1A2ALDH1A1TSHR
SCHEMBL6294025 0.76 PARP1 (0.46) PARP1DAOMEN1CYP1A2KMT2A
SCHEMBL6804934 0.76 CYP1A2 (0.65) MEN1CYP1A2KMT2AALDH1A1TSHR
SCHEMBL6794703 0.75 PARP1 (0.46) PARP1DAOPARP2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6872727-B1 Polycyclic pyrimidine -2,4(1H,3H)-diones with functionalized alkyl residues at the 1- and/or 3-position(s); methods for their synthesis and pharmaceutical preparation PRIVATES INSTITUT FUR BIOMEDIZINISCHE FORSCHUNG UND BERATUNG (DE) 2005-03-29 US disclosed
EP-1150964-B1 POLYCYCLIC PYRIMIDINE-2,4(1H, 3H)-DIONE WITH FUNCTIONALIZED ALKYL RADICALS IN 1- AND/OR 3-POSITION, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS IBFB GMBH PRIVATES INST FUER B (DE) 2003-10-29 EP disclosed
EP-1150964-A2 POLYCYCLIC PYRIMIDINE-2,4(1H, 3H)-DIONE WITH FUNCTIONALIZED ALKYL RADICALS IN 1- AND/OR 3-POSITION, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS IBFB GmbH Privates Institut für biomedizinische Forschung und Beratung (DE) 2001-11-07 EP disclosed
WO-2001014344-A2 POLYCYCLIC PYRIMIDINE-2,4(1H, 3H)-DIONE WITH FUNCTIONALIZED ALKYL RADICALS IN 1- AND/OR 3-POSITION, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS IBFB GMBH PRIVATES INSTITUT FÜR BIOMEDIZINISCHE FORSCHUNG UND BERATUNG (DE) 2001-03-01 WO disclosed