SCHEMBL1724355

SCHEMBL1724355

OB(O)c1cccc(CN2CCCC2)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.60
ALDH1A1 P00352 2/20 0.60
PRMT6 Q96LA8 1/20 0.57
TDP1 Q9NUW8 1/20 0.56
ENPP2 Q13822 2/20 0.55
CYP2D6 P10635 2/20 0.54
CYP2C9 P11712 1/20 0.54
HIF1A Q16665 1/20 0.54
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.51
CYP2C19 P33261 1/20 0.47
HRH3 Q9Y5N1 3/20 0.47
LPL P06858 2/20 0.46
LIPG Q9Y5X9 2/20 0.46
MBTD1 Q05BQ5 1/20 0.46
TP53BP1 Q12888 1/20 0.46
L3MBTL3 Q96JM7 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL29955383 0.98 SMN1; SMN2 (0.58) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
SCHEMBL2248354 0.98 SMN1; SMN2 (0.63) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
SCHEMBL29955283 0.98 SMN1; SMN2 (0.63) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
Hydrochloric Acid SCHEMBL29950873 0.97 SMN1; SMN2 (0.61) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
Hydrochloric Acid SCHEMBL2279012 0.97 SMN1; SMN2 (0.61) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
SCHEMBL2561398 0.87 NCF1 (0.55) SMN1; SMN2ALDH1A1PRMT6TDP1ENPP2
SCHEMBL3666137 0.85 MC4R (0.57) SMN1; SMN2ALDH1A1PRMT6ENPP2KDM4E
SCHEMBL875822 0.85 NCF1 (0.60) SMN1; SMN2ALDH1A1ENPP2KDM4EHRH3
SCHEMBL16633728 0.84 L3MBTL3 (0.64) SMN1; SMN2ALDH1A1TDP1ENPP2CYP2D6
Hydrochloric Acid SCHEMBL29952963 0.84 NCF1 (0.59) SMN1; SMN2ALDH1A1ENPP2KDM4EHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403833-A1 8-SUBSTITUTED QUINOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2012-01-11 EP disclosed
WO-2010101949-A1 8-SUBSTITUTED QUINOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2010-09-10 WO disclosed
WO-2010101949-A1 8-SUBSTITUTED QUINOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2010-09-10 WO disclosed