SCHEMBL17244337

SCHEMBL17244337

COc1ccc(-c2nc(N)c3cc(OC)ccc3c2N=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.41
ADORA2A P29274 1/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
SYK P43405 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
KMT2A Q03164 1/20 0.40
ADORA1 P30542 1/20 0.40
PLAU P00749 1/20 0.39
DYRK1A Q13627 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
MAP4K4 O95819 1/20 0.38
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2429295 0.76 MAPT (0.43) DHFRADORA2ASYKMAPTSMN1; SMN2
SCHEMBL5199692 0.69 MAPT (0.51) MAPTSMN1; SMN2KMT2ADYRK1APDE3B
SCHEMBL6700778 0.67 KMT2A (0.54) DHFRADORA2AMAPTSMN1; SMN2KMT2A
SCHEMBL2425567 0.66 NPC1 (0.53) ADORA2ASYKMAPTCYP1A2KMT2A
SCHEMBL12076878 0.65 CYP1A1 (0.56) ADORA2AMAPTSMN1; SMN2CYP1A1CYP1A2
SCHEMBL11087367 0.65 APOBEC3A (0.47) APOBEC3AAPOBEC3GMAPTSMN1; SMN2CYP1A2
SCHEMBL21852751 0.64 ALDH1A1 (0.67) ADORA2AMAPTKMT2AADORA1CA1
SCHEMBL11086899 0.64 APOBEC3A (0.42) APOBEC3AAPOBEC3GMAPTSMN1; SMN2CYP1A2
SCHEMBL1622459 0.64 KDM4E (0.54) MAPTSMN1; SMN2CYP1A2KMT2ADYRK1A
SCHEMBL4124300 0.64 ENPP1 (0.66) KMT2ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542239-B1 USE OF ISOQUINOLONES FOR PREPARING DRUGS, NOVEL ISOQUINOLONES AND METHOD FOR SYNTHESISING SAME Université Joseph Fourier (FR) 2015-11-11 EP disclosed