SCHEMBL1724945

SCHEMBL1724945

C=Cc1cnn(C(=O)O)c(=O)c1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.36
PTGS2 P35354 1/20 0.33
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9988990 0.69 IDH1 (0.39)
SCHEMBL34470588 0.67 CNR2 (0.38)
SCHEMBL28191634 0.60 HCAR2 (0.52) PTGS2
SCHEMBL29955798 0.60 HCAR2 (0.52) PTGS2
SCHEMBL9316209 0.58 PARP1 (0.42) PTGS2PARP1
SCHEMBL6774970 0.57 NAPRT (0.44) PTGS1PTGS2PARP1
SCHEMBL6551393 0.57 HDAC8 (0.46) PTGS2PARP1
SCHEMBL28500105 0.57 HTT (0.49)
SCHEMBL20876169 0.56 ALOX15 (0.54) PARP1
SCHEMBL30108195 0.56 RAF1 (0.53) PTGS2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406233-A1 AZA PYRIDONE ANALOGS USEFUL AS MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS Bristol-Myers Squibb Company (US) 2012-01-18 EP disclosed
WO-2010104818-A1 AZA PYRIDONE ANALOGS USEFUL AS MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-09-16 WO disclosed