SCHEMBL1725979

SCHEMBL1725979

Cc1nn(C)c(O)c1-c1c(F)cc(F)cc1F.Cc1nn(C)c(Oc2c(F)cc([N+](=O)[O-])cc2F)c1-c1c(F)cc(F)cc1F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.38
DAPK3 O43293 1/20 0.38
GRK5 P34947 1/20 0.38
LIMK1 P53667 1/20 0.38
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1725765 0.94 CHEK1 (0.42) CHEK1DAPK3GRK5LIMK1MAPT
SCHEMBL170898 0.76 PDE10A (0.34) MAPTL3MBTL1CYP1A2CYP3A4CYP2C9
SCHEMBL1727361 0.76 CYP1A2 (0.32) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL170955 0.73 POLB (0.35) CYP1A2CYP3A4CYP2C9CYP2C19POLB
SCHEMBL1724939 0.67 PDE10A (0.41) MAPTSMN1; SMN2CYP1A2CYP3A4CYP2C9
SCHEMBL1724913 0.66 PDE2A (0.41) LMNACYP1A2POLB
SCHEMBL22143978 0.65 MAPT (0.48) CHEK1DAPK3GRK5LIMK1MAPT
SCHEMBL27212602 0.63 PKM (0.47) CHEK1DAPK3GRK5LIMK1MAPT
SCHEMBL13106292 0.63 CHEK1 (0.51) CHEK1DAPK3GRK5LIMK1MAPT
SCHEMBL10751685 0.61 CHEK1 (0.49) CHEK1DAPK3GRK5LIMK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403834-A1 Fungicidal pyrazoles E. I. du Pont de Nemours and Company (US) 2012-01-11 EP disclosed
WO-2010101973-A1 FUNGICIDAL PYRAZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-09-10 WO disclosed