SCHEMBL172624

SCHEMBL172624

CCCC(NC)c1cccc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.48
TAS1R1 Q7RTX1 1/20 0.48
PNMT P11086 1/20 0.46
SLC6A4 P31645 2/20 0.44
SLC6A2 P23975 1/20 0.44
EPHX1 P07099 1/20 0.44
HTR2A P28223 2/20 0.42
HTR2B P41595 2/20 0.42
SIGMAR1 Q99720 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
ADRA2C P18825 1/20 0.42
ADRA1A P35348 1/20 0.42
DRD3 P35462 1/20 0.42
OPRK1 P41145 1/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11065022 0.87 PNMT (0.49) PNMTSLC6A4SLC6A2HTR2AHTR2B
SCHEMBL18255649 0.87 PNMT (0.49) PNMTSLC6A4SLC6A2HTR2AHTR2B
SCHEMBL11407610 0.83 PNMT (0.47) PNMTSLC6A4SLC6A2HTR2AHTR2B
SCHEMBL10217243 0.83 PNMT (0.51) PNMTSLC6A4SLC6A2ALDH1A1POLB
SCHEMBL14262202 0.83 PNMT (0.51) PNMTSLC6A4SLC6A2ALDH1A1POLB
Hydrochloric Acid SCHEMBL19244848 0.81 PNMT (0.50) PNMTSLC6A4SLC6A2EPHX1ALDH1A1
SCHEMBL23892009 0.80 PDE2A (0.41) SLC6A4SLC6A2HTR2AHTR2BSIGMAR1
SCHEMBL19541914 0.80 PNMT (0.51) TAS1R3TAS1R1PNMTSLC6A4EPHX1
SCHEMBL18593504 0.80 PNMT (0.45) PNMTSLC6A4SLC6A2HTR2AHTR2B
SCHEMBL7929105 0.79 PNMT (0.50) TAS1R3TAS1R1PNMTSLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed