SCHEMBL1726378

SCHEMBL1726378

CS(=O)(=O)C1(S(C)(=O)=O)OB(c2cc(F)c(N)cc2F)OC1(S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.31

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL59040 0.78 LPL (0.37)
SCHEMBL29385065 0.78 LPL (0.37)
SCHEMBL2934443 0.78 PIK3R1 (0.38)
SCHEMBL23751788 0.73 CA1 (0.33) CA12CA1CA2CA4CA6
SCHEMBL15289502 0.71 LPL (0.37)
SCHEMBL19668082 0.69 LPL (0.38) CA12CA1CA2CA4CA6
SCHEMBL22397836 0.68 EGFR (0.35) CA12CA1CA2CA4CA6
SCHEMBL10278788 0.68
SCHEMBL26674620 0.66 LPL (0.38) CA12CA1CA2CA4CA6
SCHEMBL58364 0.66 LPL (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406258-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS Cellzome Limited (GB) 2012-01-18 EP disclosed
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed