SCHEMBL2934443

SCHEMBL2934443

CS(=O)(=O)C1(S(C)(=O)=O)OB(c2cnc(N)cc2F)OC1(S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 4/20 0.38
PIK3CA P42336 4/20 0.38
PIK3CD O00329 2/20 0.35
PIK3CB P42338 2/20 0.35
MTOR P42345 2/20 0.35
PIK3CG P48736 2/20 0.35
ALOX5AP P20292 2/20 0.30
FEN1 P39748 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2814938 0.80 LPL (0.34)
SCHEMBL1726378 0.78 CA12 (0.31)
SCHEMBL10328173 0.70
SCHEMBL16055897 0.66 MAP3K12 (0.36) PIK3R1PIK3CAPIK3CDPIK3CBMTOR
SCHEMBL21828795 0.66 ABL1 (0.35) PIK3CAMTOR
SCHEMBL22397836 0.65 EGFR (0.35)
SCHEMBL13016581 0.64 NOS3 (0.35)
SCHEMBL30736300 0.63 NOS3 (0.47) PIK3R1PIK3CAMTOR
SCHEMBL13089602 0.63 NOS3 (0.47) PIK3R1PIK3CAMTOR
SCHEMBL20519666 0.63 NOS3 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984350-B1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS NOVARTIS AG (CH) 2010-08-18 EP disclosed