SCHEMBL172705

SCHEMBL172705

CCC[C@@H](COCc1ccccc1)NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.46
BCHE P06276 1/20 0.43
TSHR P16473 1/20 0.42
SIGMAR1 Q99720 2/20 0.42
CA1 P00915 4/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
FOLH1 Q04609 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27803762 0.83 SIGMAR1 (0.52) SIGMAR1
Hydrochloric Acid SCHEMBL10756071 0.81 SIGMAR1 (0.50) SIGMAR1
SCHEMBL13995917 0.81 TACR1 (0.46) TACR1BCHETSHRSIGMAR1CA1
SCHEMBL7265738 0.81 CA1 (0.47) TACR1TSHRCA1CA2CA7
SCHEMBL12018717 0.81 CA1 (0.47) TACR1TSHRCA1CA2CA7
SCHEMBL7265733 0.81 CA1 (0.47) TACR1TSHRCA1CA2CA7
SCHEMBL21755741 0.80 SIGMAR1 (0.49) SIGMAR1
SCHEMBL6119036 0.79 FOLH1 (0.48) TACR1CA1CA2CA7CA9
SCHEMBL8327295 0.79 IDO1 (0.40) TACR1BCHE
SCHEMBL15341689 0.78 BCHE (0.43) TACR1BCHETSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed