SCHEMBL1727178

SCHEMBL1727178

COc1cc2nc(-c3cccc(NC(=O)CN4CCOCC4)c3)nc(Nc3ccc4[nH]ncc4c3)c2cc1O

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.81
ROCK1 Q13464 5/20 0.62
PRKD3 O94806 2/20 0.56
CSNK2A1 P68400 2/20 0.56
STK3 Q13188 2/20 0.56
AURKB Q96GD4 2/20 0.56
CLK4 Q9HAZ1 2/20 0.56
STK17A Q9UEE5 2/20 0.56
PLK4 O00444 1/20 0.56
CHEK2 O96017 1/20 0.56
PRKCG P05129 1/20 0.56
PHKG2 P15735 1/20 0.56
CDK2 P24941 1/20 0.56
AKT1 P31749 1/20 0.56
AKT2 P31751 1/20 0.56
MAP2K2 P36507 1/20 0.56
PRKCI P41743 1/20 0.56
MAPKAPK2 P49137 1/20 0.56
PRKCQ Q04759 1/20 0.56
ACVR1 Q04771 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1722249 0.91 ROCK2 (0.87) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL1724850 0.89 ROCK2 (1.00) ROCK2ROCK1PRKD3CSNK2A1STK3
Trifluoroacetic Acid SCHEMBL1723799 0.87 ROCK2 (0.81) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL876581 0.87 ROCK2 (0.70) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL3795144 0.85 ROCK2 (0.61) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL11919876 0.85 PRKD3 (0.77) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL877371 0.85 ROCK2 (1.00) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL3798011 0.83 ROCK2 (0.58) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL20953095 0.82 ROCK2 (0.67) ROCK2ROCK1PRKD3CSNK2A1STK3
SCHEMBL20953067 0.82 ROCK2 (0.67) ROCK2ROCK1PRKD3CSNK2A1STK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406236-A1 RHO KINASE INHIBITORS Surface Logix, Inc. (US) 2012-01-18 EP disclosed
WO-2010104851-A1 RHO KINASE INHIBITORS SURFACE LOGIX, INC. (US) 2010-09-16 WO disclosed