SCHEMBL17276804

SCHEMBL17276804

CC(C)[C@H]1C(=O)c2cc(-c3ccc(C(=O)O)cc3)ccc2OC12CCNCC2

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 9/20 0.43
KCNH2 Q12809 7/20 0.41
CYP2D6 P10635 6/20 0.41
TDP2 O95551 1/20 0.37
RARB P10826 7/20 0.37
RARG P13631 7/20 0.37
RXRA P19793 4/20 0.37
RARA P10276 7/20 0.36
OPRK1 P41145 5/20 0.36
RXRB P28702 2/20 0.35
RXRG P48443 1/20 0.35
OPRM1 P35372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17276900 0.79 CYP2D6 (0.39) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL17276832 0.79 CYP2D6 (0.39) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL3837866 0.74 OPRD1 (0.42) OPRD1KCNH2CYP2D6TDP2RXRA
SCHEMBL3836335 0.70 OPRD1 (0.36) OPRD1KCNH2CYP2D6TDP2RARG
Hydrochloric Acid SCHEMBL1814403 0.70 OPRD1 (0.36) OPRD1KCNH2CYP2D6TDP2RARB
SCHEMBL4272876 0.67 TP53 (0.35) OPRD1KCNH2RARBOPRK1
SCHEMBL1823244 0.67 BACE1 (0.42) OPRD1
SCHEMBL12761461 0.66 HDAC3 (0.54) OPRD1KCNH2CYP2D6OPRK1OPRM1
SCHEMBL17276802 0.66 HDAC3 (0.50)
SCHEMBL16334838 0.66 IL2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145933-A1 NAMPT INHIBITORS AND METHODS Genzyme Corporation (US) 2017-03-29 EP disclosed
WO-2015179759-A1 NAMPT INHIBITORS AND METHODS GENZYME CORPORATION (US) 2015-11-26 WO disclosed