SCHEMBL4272876

SCHEMBL4272876

CCCCOC(=O)C1C(=O)c2cc(C(=O)O)ccc2OC12CCNCC2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
CNR2 P34972 2/20 0.35
PLA2G4B P0C869 1/20 0.34
OPRD1 P41143 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RARB P10826 3/20 0.33
HTT P42858 1/20 0.33
OPRK1 P41145 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739214 0.92 HPGD (0.32) TP53TSHRCNR2OPRD1MEN1
SCHEMBL7845728 0.85 OPRD1 (0.38) TSHROPRD1OPRK1KCNH2
SCHEMBL3836335 0.82 OPRD1 (0.36) CNR2OPRD1ALDH1A1OPRK1KCNH2
SCHEMBL7849699 0.79 AGTR2 (0.42)
SCHEMBL7852250 0.79 HPGD (0.40) TP53MEN1KMT2AKDM4EALDH1A1
SCHEMBL7843937 0.78 NR3C1 (0.36) TP53MEN1KMT2AKDM4EALDH1A1
SCHEMBL3837866 0.77 OPRD1 (0.42) CNR2OPRD1ALDH1A1OPRK1KCNH2
SCHEMBL2594953 0.71 GAA (0.43) TSHROPRD1OPRK1KCNH2
SCHEMBL4272883 0.70 HDAC3 (0.46) KMT2AKDM4EALDH1A1HPGDHTT
SCHEMBL4708596 0.70 ACACA (0.36) TP53OPRD1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed