SCHEMBL1728577

SCHEMBL1728577

O=C(O)NCCN1CCN(c2cccc3ccccc23)CC1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.67
DRD3 P35462 7/20 0.67
HTR1A P08908 6/20 0.67
HTR2A P28223 3/20 0.67
HTR2C P28335 3/20 0.67
DRD4 P21917 3/20 0.63
FAAH O00519 1/20 0.53
CNR1 P21554 1/20 0.53
SLC6A4 P31645 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727824 0.92 DRD3 (0.75) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL1728118 0.85 DRD3 (0.59) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL23751044 0.82 MEN1 (0.62) DRD4FAAH
SCHEMBL4513849 0.81 DRD3 (1.00) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL239772 0.80 DRD4 (0.58) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL3664190 0.79 DRD2 (0.59) DRD2DRD3HTR1AHTR2AHTR2C
Hydrochloric Acid SCHEMBL237609 0.79 DRD4 (0.57) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL9283836 0.79 DRD2 (0.59) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL23750995 0.79 HSD17B10 (0.64) DRD2DRD3HTR1ADRD4
SCHEMBL13711982 0.77 DRD3 (0.60) DRD2DRD3HTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP disclosed
CN-1812980-B Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their use as pharmaceuticals SANOFI AVENTIS 2011-04-06 CN disclosed
CN-101712660-A Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their therapeutic use SANOFI AVENTIS 2010-05-26 CN disclosed
CN-1812980-A Piperidinyl-and piperazinyl-alkylcarbamate derivatives, their preparation and their therapeutic use SANOFI AVENTIS (FR) 2006-08-02 CN disclosed
EP-1633735-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS Sanofi-Aventis (FR) 2006-03-15 EP disclosed
WO-2004099176-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI-AVENTIS (FR) 2004-11-18 WO disclosed