SCHEMBL1728599

SCHEMBL1728599

Fc1ccc(-c2cn3ccsc3n2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 10/20 0.66
NPC1 O15118 9/20 0.66
RAB9A P51151 9/20 0.66
MAPT P10636 5/20 0.66
NFKB1 P19838 4/20 0.66
NFKB2 Q00653 4/20 0.66
RELA Q04206 4/20 0.66
TP53 P04637 14/20 0.59
LMNA P02545 2/20 0.56
ALOX15 P16050 2/20 0.56
POLB P06746 2/20 0.56
MEN1 O00255 1/20 0.56
MAPK1 P28482 1/20 0.56
KMT2A Q03164 1/20 0.56
HPGD P15428 3/20 0.56
ALDH1A1 P00352 2/20 0.56
HSD17B10 Q99714 2/20 0.56
ALOX12 P18054 1/20 0.56
TSHR P16473 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12970198 0.83 NPC1 (0.66) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL1692138 0.83 NPC1 (0.66) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL12692485 0.83 SMN1; SMN2 (0.70) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL4147815 0.83 NPC1 (0.66) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL969616 0.83 NPC1 (0.66) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL30059210 0.83 NPC1 (0.66) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL5773733 0.83 TP53 (0.68) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL2496897 0.83 TP53 (0.68) SMN1; SMN2NPC1RAB9AMAPTNFKB1
Bromide SCHEMBL3869607 0.82 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL4781521 0.80 NPC1 (0.61) SMN1; SMN2NPC1RAB9AMAPTNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115323409-B Method for electrochemically synthesizing asymmetric double heteroaromatic compounds 南京工业大学 2025-05-23 CN disclosed
CN-115323409-A Method for electrochemically synthesizing asymmetric double-hetero aromatic hydrocarbon compound 南京工业大学 2022-11-11 CN disclosed
US-20210299131-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NATIONAL INSTITUTES OF HEALTH 2021-09-30 US disclosed
US-10953017-B2 Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such SOUTHERN RESEARCH INSTITUTE (US) 2021-03-23 US disclosed
US-20200171040-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH SOUTHERN RES INST (US) 2020-06-04 US disclosed
US-20190083505-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NATIONAL INSTITUTES OF HEALTH 2019-03-21 US disclosed
US-9980969-B2 Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such SOUTHERN RESEARCH INSTITUTE (US) 2018-05-29 US disclosed
US-9980969-B2 Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such SOUTHERN RESEARCH INSTITUTE (US) 2018-05-29 US disclosed
US-20160022691-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH SOUTHERN RES INST (US) 2016-01-28 US disclosed
US-20160022691-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH SOUTHERN RES INST (US) 2016-01-28 US disclosed
US-20080161341-A1 Novel imidazothiazoles and imidazoxazoles ABBVIE INC. 2008-07-03 US disclosed
US-20080161341-A1 Novel imidazothiazoles and imidazoxazoles ABBVIE INC. 2008-07-03 US disclosed
WO-2008063287-A2 NOVEL IMIDAZOTHIAZOLES AND IMIDAZOXAZOLES ABBOTT LABORATORIES (US) 2008-05-29 WO disclosed
US-20070270418-A1 Inhibitors of P38 and Methods of Using the Same ARQULE, INC. 2007-11-22 US disclosed
US-20070270418-A1 Inhibitors of P38 and Methods of Using the Same ARQULE, INC. 2007-11-22 US disclosed
US-20070270418-A1 Inhibitors of P38 and Methods of Using the Same ARQULE, INC. 2007-11-22 US disclosed
EP-1809636-A1 SYNTHESIS OF IMIDAZOOXAZOLE AND IMIDAZOTHIAZOLE INHIBITORS OF P38 MAP KINASE ARQULE, INC. (US) 2007-07-25 EP disclosed
WO-2006044869-A1 SYNTHESIS OF IMIDAZOOXAZOLE AND IMIDAZOTHIAZOLE INHIBITORS OF P38 MAP KINASE ARQULE, INC. (US) 2006-04-27 WO disclosed
EP-1633758-A2 IMIDAZOTHIAZOLES AND IMIDAZOXAZOLE DERIVATIVES AS INHIBITORS OF P38 ARQULE, INC. (US) 2006-03-15 EP disclosed
WO-2004110990-A2 IMIDAZOTHIAZOLES AND IMIDAZOXAZOLE DERIVATIVES AS INHIBITORS OF P38 ARQULE, INC. (US) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160022691-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NFKBIA, NFRKB, TFEB SMN1; SMN2 33/4885NPC1 489/4885RAB9A 2424/4885
US-20200171040-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NFKBIA, NFRKB, TFEB SMN1; SMN2 29/4885NPC1 467/4885RAB9A 2402/4885
US-20190083505-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NFKBIA, NFRKB, TFEB SMN1; SMN2 29/4885NPC1 467/4885RAB9A 2402/4885
US-20070270418-A1 Inhibitors of P38 and Methods of Using the Same MAPK1, MAPK8, MAPK7 SMN1; SMN2 2415/4885NPC1 2774/4885RAB9A 1851/4885
US-20080161341-A1 Novel imidazothiazoles and imidazoxazoles MAP3K1, MAP3K19, MAP3K5 SMN1; SMN2 3838/4885NPC1 2227/4885RAB9A 3058/4885
US-20210299131-A1 TREATMENT OF NEURODEGENERATIVE DISEASES, CAUSATION OF MEMORY ENHANCEMENT, AND ASSAY FOR SCREENING COMPOUNDS FOR SUCH NFKBIA, NFRKB, TFEB SMN1; SMN2 29/4885NPC1 467/4885RAB9A 2402/4885
US-10953017-B2 Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such NFKBIA, NFRKB, TFEB SMN1; SMN2 29/4885NPC1 467/4885RAB9A 2402/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.