SCHEMBL1729490

SCHEMBL1729490

Cc1ccc(Oc2ccc(-n3ccn(-c4ccc(OCCN(C)C)cc4)c3=O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.56
LTA4H P09960 2/20 0.52
MCHR1 Q99705 2/20 0.51
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
HRH3 Q9Y5N1 2/20 0.43
KCNH2 Q12809 2/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728669 0.90 LTA4H (0.68) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL1728621 0.89 MCHR1 (0.63) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL1727319 0.88 LTA4H (0.51) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL1727854 0.88 LTA4H (0.52) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL6081522 0.85 ALDH1A1 (0.55) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL6080985 0.85 MCHR1 (0.54) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL6081903 0.85 MCHR1 (0.54) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL1728515 0.84 MCHR1 (0.52) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL6081331 0.84 MCHR1 (0.53) MAPK14LTA4HMCHR1CYP1A2CYP2D6
SCHEMBL1728477 0.84 MCHR1 (0.56) MAPK14MCHR1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551810-B1 DIARYL-SUBSTITUTED CYCLIC UREA DERIVATIVES HAVING AN MCH-MODULATORY EFFECT SANOFI AVENTIS DEUTSCHLAND (DE) 2011-11-30 EP disclosed
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed