SCHEMBL17295331

SCHEMBL17295331

OCC#Cc1ccc(Br)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.42
EGFR P00533 1/20 0.37
MMP2 P08253 1/20 0.37
MMP12 P39900 1/20 0.37
ALDH1A1 P00352 1/20 0.36
P2RY6 Q15077 1/20 0.34
FFAR1 O14842 3/20 0.33
FFAR4 Q5NUL3 2/20 0.33
GRM5 P41594 1/20 0.33
KDM1A O60341 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RCOR1 Q9UKL0 1/20 0.33
KCNH2 Q12809 2/20 0.33
KDM1B Q8NB78 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
GABRP O00591 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16922697 0.85 KDM1A (0.34) FFAR1FFAR4GRM5KDM1ARCOR1
SCHEMBL81135 0.84 MELK (0.47) MELKEGFRMMP2MMP12ALDH1A1
SCHEMBL15588319 0.81 PTPN2 (0.33) EGFRMMP2MMP12FFAR1FFAR4
SCHEMBL15588338 0.80 FFAR1 (0.34) EGFRMMP2MMP12FFAR1FFAR4
SCHEMBL7651081 0.79 CYP2D6 (0.36) GRM5KDM1ACYP1A2CYP2D6CYP2C9
SCHEMBL13531864 0.78 MELK (0.42) MELKMMP2MMP12ALDH1A1P2RY6
SCHEMBL80226 0.76 KIF11 (0.47) MELKEGFRMMP2MMP12ALDH1A1
SCHEMBL7788815 0.75 FFAR1 (0.43) MMP2MMP12FFAR1FFAR4GRM5
SCHEMBL16840949 0.75 HTT (0.35) FFAR1FFAR4NPSR1KIF11
SCHEMBL19608768 0.75 CYP1A1 (0.39) EGFRGRM5KDM1ACYP1A2RCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed