SCHEMBL17295372

SCHEMBL17295372

CSc1ccc(-c2nn(C)c(O)c2C=O)cc1F.CSc1ccc(-c2nn(C)c(O)c2C=O)cc1F

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.33
STK17B O94768 1/20 0.33
AR P10275 2/20 0.33
POLB P06746 1/20 0.30
PIK3CD O00329 1/20 0.30
ABL1 P00519 1/20 0.30
EGFR P00533 1/20 0.30
HCK P08631 1/20 0.30
SRC P12931 1/20 0.30
KDR P35968 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
MTOR P42345 1/20 0.30
PIK3CG P48736 1/20 0.30
EPHB4 P54760 1/20 0.30
PRKDC P78527 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17290640 1.00 ERN1 (0.33) ERN1STK17BARPOLBPIK3CD
SCHEMBL17290263 0.85 PTGS2 (0.35) POLB
SCHEMBL17290593 0.84 COMT (0.34) ERN1
SCHEMBL17290381 0.83 ERN1 (0.36) ERN1POLBPIK3CDABL1EGFR
SCHEMBL17290446 0.82 GRM5 (0.34) STK17BARPOLBPIK3CDABL1
SCHEMBL17290345 0.80 ERN1 (0.50) ERN1PIK3CDABL1EGFRHCK
SCHEMBL17295073 0.79 ALDH1A1 (0.40) POLB
SCHEMBL17290566 0.79 ALDH1A1 (0.40) POLB
SCHEMBL17290537 0.78 MAPK14 (0.41) ARPOLB
SCHEMBL17290229 0.77 POLB (0.36) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3148972-A1 PYRAZOLONE DERIVATIVES AS NITROXYL DONORS Cardioxyl Pharmaceuticals Inc. (US) 2017-04-05 EP disclosed
WO-2015183839-A1 PYRAZOLONE DERIVATIVES AS NITROXYL DONORS CARDIOXYL PHARMACEUTICALS, INC. (US) 2015-12-03 WO disclosed